Evigrade
Major

citalopram × tacrolimus

SSRI (selective serotonin reuptake inhibitor)×Calcineurin inhibitor (immunosuppressant)

Mechanism

Tacrolimus prolongs the QT interval, especially with hypomagnesaemia (common on calcineurin inhibitors). Citalopram also prolongs QT dose-dependently (FDA caps at 40 mg/day). Effects add up.

Symptoms

QT prolongation on ECG, dizziness, syncope, palpitations. Severe cases: polymorphic ventricular tachycardia (torsades de pointes). Risk rises with hypokalaemia and hypomagnesaemia.

Management

Avoid the combination. Alternative antidepressants with minimal QT effect post-transplant: mirtazapine, agomelatine, sertraline (up to 100 mg/day). ECG before start and at 2 weeks; maintain potassium and magnesium.

Sources

All interactions