Evigrade
Major

Amiodarone × citalopram

Class III antiarrhythmics (Vaughan Williams)×SSRI (selective serotonin reuptake inhibitor)

Mechanism

Dual QT-prolongation risk. Citalopram carries an FDA boxed warning about dose-dependent QT effect (FDA Celexa caps at 40 mg/day); amiodarone is a potent QT-prolonging drug.

Symptoms

QT prolongation on ECG. Clinically: dizziness, syncope, palpitations. Severe cases progress to polymorphic ventricular tachycardia (torsades de pointes). Risk is higher with hypokalaemia, hypomagnesaemia, bradycardia, and ischaemic heart disease.

Management

Avoid the combination. Alternative antidepressants: mirtazapine or agomelatine (minimal QT effect). If citalopram is needed, cap at 20 mg/day; ECG before start and at 2 weeks.

Sources

All interactions

Amiodarone and citalopram: interaction, management, sources – Evigrade