Evigrade
Minor

Amitriptyline × Spironolactone

Tricyclic antidepressants (TCA)×Potassium-sparing diuretics (mineralocorticoid receptor antagonists)

Mechanism

No direct interaction. Additive orthostatic hypotension possible in older patients during hypovolaemia: spironolactone via diuresis, amitriptyline via α1-blockade.

Symptoms

Possible postural dizziness, fatigue. In older patients: fall risk.

Management

Begin amitriptyline at 10 mg at bedtime. In older patients, do not exceed 25 mg/day. Check standing/sitting BP at 1–2 weeks. With pronounced orthostatic hypotension, consider neuropathic-pain alternatives: gabapentin or pregabalin.

Sources

All interactions