Evigrade
Moderate

Amitriptyline × Nitroglycerin

Tricyclic antidepressants (TCA)×Organic nitrate

Mechanism

Additive orthostatic hypotension with sublingual nitroglycerin. Amitriptyline blocks α1-adrenoceptors and reduces compensatory response.

Symptoms

Postural dizziness, syncope, fatigue. Older patients: fall and fracture risk.

Management

The patient takes the first nitroglycerin dose sitting or lying down. Older patients: enhanced fall monitoring. Alternative antidepressants without α1-blockade: sertraline or agomelatine.

Sources

All interactions