Evigrade
Moderate

Amitriptyline × Glibenclamide

Tricyclic antidepressants (TCA)×Oral hypoglycemic agents. Sulfonylureas

Mechanism

TCAs may mask hypoglycaemia symptoms (tremor, tachycardia) via anticholinergic effect. No direct pharmacokinetic interaction.

Symptoms

Sudden confusion, weakness, ataxia without preceding tachycardia or sweating. Older patients: risk of severe hypoglycaemia without warning symptoms.

Management

Warn the patient that the TCA masks hypoglycaemia warning signs. Check glucose more often (4 times daily in the first week, then by self-monitoring). In older patients, prefer gliclazide (less hypoglycaemia) or metformin/DPP-4 inhibitor over glibenclamide.

Sources

All interactions